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Targets Recommended: Others

7

抑制剂 & 化合物

1

天然产物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T0382 Eprodisate disodium

NC-503,伊罗地塞二钠,伊罗地塞二钠盐

Others Others
Eprodisate disodium (NC-503) 是一种带负电荷的磺化类的原纤维形成抑制剂,是口服具有活力的 Eprodisate 二钠盐形式,可用于研究淀粉样蛋白A(AA) 淀粉样变性病。
T31527 Disalicylalpropylenediimine

Disalicylalpropylenediimine is a biochemical.
T37851 Chlorido[N,N'-disalicylidene-1,2-phenylenediamine]iron(III)

Chlorido[N,N'-disalicylidene-1,2-phenylenediamine]iron(III) is an inducer of ferroptosis.1 It induces ferroptosis, but not apoptosis or necroptosis, in NB1 cancer cells when used at a concentration of 3 μM.1 Chlorido[N,N'-disalicylidene-1,2-phenylenediamine]iron(III) inhibits proliferation of BJAB, NALM-6, Jurkat, MelHO, and MCF-7 cancer cells (IC50s = 0.07, 2.5, 1.5, 3, and 5 μM, respectively), as well as NALM-6 cells resistant to daunorubicin and vincristine when used at concentrations ranging...
T39638 Eprodisate

Eprodisate is a novel compound specifically developed to disrupt the interactions between amyloidogenic proteins and glycosaminoglycans, effectively impeding the polymerization of amyloid fibrils and their deposition in tissues. This compound shows potential for delaying the advancement of AA amyloidosis-related renal disease and could apply to various forms of amyloidosis.
T24863 Tedisamil

Tedisamilum,Pulzium

Tedisamil is a blocker of K+ currents in cardiac tissues, exerts bradycardic effects. It is an antiarrhythmic drug with predominantly class III activity. It has shown clinical efficacy in angina pectoris.
T70524 Tedisamil sesquifumarate

Tedisamil sesquifumarate is an Antiarrhythmic Agent (K(sup +) Channel Blocker)
T71874 ST056083

ST056083 is an inhibitor of the c-di-AMP synthetase DNA integrity scanning protein (DisA) in vitro.

化合物

Eprodisate disodium
Cat.No: T0382
Synonym: NC-503,伊罗地塞二钠,伊罗地塞二钠盐
Target: Others
Disalicylalpropylenediimine
Cat.No: T31527
Synonym:
Target:
Chlorido[N,N'-disalicylidene-1,2-phenylenediamine]iron(III)
Cat.No: T37851
Synonym:
Target:
Eprodisate
Cat.No: T39638
Synonym:
Target:
Tedisamil
Cat.No: T24863
Synonym: Tedisamilum,Pulzium
Target:
Tedisamil sesquifumarate
Cat.No: T70524
Synonym:
Target:
ST056083
Cat.No: T71874
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T83564 (2E,4E)-8-Hydroxy-2,7-dimethyl-decadien-(2,4)-disaeure-(1,10)-dioic acid

'(2E,4E)-8-Hydroxy-2,7-dimethyl-decadien-(2,4)-disaeure-(1,10)-dioic acid',作为一种从木耳花中分离得到的天然产物,展现出抗氧化和抗炎的活性。

天然产物

(2E,4E)-8-Hydroxy-2,7-dimethyl-decadien-(2,4)-disaeure-(1,10)-dioic acid
Cat.No: T83564
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPH-02993 DisA Protein, Mycobacterium paratuberculosis, Recombinant (His & Myc)

disA,c-di-AMP synthase,DNA integrity scanning prote...

Mycobacterium paratuberculosis E. coli
Participates in a DNA-damage check-point. DisA forms globular foci that rapidly scan along the chromosomes searching for lesions.; Has also diadenylate cyclase activity, catalyzing the condensation of 2 ATP molecules into cyclic di-AMP (c-di-AMP). c-di-AMP likely acts as a signaling molecule that may couple DNA integrity with a cellular process. DisA Protein, Mycobacterium paratuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predict...

重组蛋白

DisA Protein, Mycobacterium paratuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-02993
Species: Mycobacterium paratuberculosis
Expression System: E. coli
TargetMol Loading
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