Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80137 |
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
d(CH2)5[Tyr(Me)2, Dab5]AVP |
Vasopressin Receptor | GPCR/G Protein |
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP)作为针对加压素受体V1a的特异性拮抗剂,具有pA2值为6.71。 |