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39

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1545L1	FFAGLDD amine salt	Others	Others
	FFAGLDD amine salt 是MMP9选择性裂解肽，用于多柔比星（DOX）的胞浆递送，实现时间和空间可控的缓慢药物递送和释放。
T17946	Fmoc-Ala-Ala-Asn(Trt)-OH	Others	Others
	Fmoc-Ala-Ala-Asn(Trt)-OH 是一种可切割的 ADC 接头，用于抗体-药物偶联物。
T4271	Diroximel fumarate Diroximel Fumarete	Others	Others
	Diroximel fumarate (Diroximel Fumarete) 是一种控释制剂，是口服具有活力的富马酸单乙酯的前体药物。它被认为与其活性代谢物富马酸二甲酯的活性等效。它具有良好的安全性和有效性，具有研究多发性硬化的潜力。
T14724	Boc-Cystamine	Others	Others
	Boc-Cystamine is a cleavable linker vital in ADC synthesis. Boc-Cystamine joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T40762	NO2-SPDB-sulfo NO2-SPDB-sulfo
	NO2-SPDB-sulfo is a cleavable linker vital in ADC synthesis. NO2-SPDB-sulfo joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T18786	TCO-SS-amine	Others	Others
	TCO-SS-amine is a cleavable linker vital in ADC synthesis. TCO-SS-amine joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T17812	DBCO-SS-amine	Others	Others
	DBCO-SS-amine is a cleavable linker vital in ADC synthesis. DBCO-SS-amine joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T17836	DMAC-SPP	Others	Others
	DMAC-SPP is a cleavable linker vital in ADC synthesis. DMAC-SPP joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T18559	PPC-NHS ester 2,5-Dioxopyrrolidin-1-yl 3-(pyridin-2-yldisulfanyl)butanoate	Others	Others
	PPC-NHS ester is a cleavable linker vital in ADC synthesis. PPC-NHS ester joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T17540	BCN-SS-NHS	Others	Others
	BCN-SS-NHS is a cleavable linker vital in ADC synthesis. BCN-SS-NHS joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T15927	m-PEG8-Amine	Others	Others
	m-PEG8-Amine is a cleavable linker vital in ADC synthesis. m-PEG8-Amine joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T39538	BCOT-PEF3-OPFP BCOT-PEF3-OPFP
	BCOT-PEF3-OPFP is a cleavable linker vital in ADC synthesis. BCOT-PEF3-OPFP joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T17524	Azidoethyl-SS-propionic acid	Others	Others
	Azidoethyl-SS-propionic acid is an ADC linker, specifically designed for the synthesis of antibody-drug conjugates (ADCs)[1]. It possesses cleavable properties, allowing for the controlled release of drug payloads.
T39169	Tetrazine-biotin
	Tetrazine-biotin is a cleavable linker vital in ADC synthesis. Tetrazine-biotin joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T40764	DMAC-SPDB
	DMAC-SPDB is a cleavable linker vital in ADC synthesis. DMAC-SPDB joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T18732	sulfo-SPDB	Others	Others
	sulfo-SPDB is a cleavable linker vital in ADC synthesis. sulfo-SPDB joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T18505	NO2-SPDMV	Others	Others
	NO2-SPDMV is a cleavable linker vital in ADC synthesis. NO2-SPDMV joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T38597	SPDP-sulfo
	SPDP-sulfo is a cleavable linker vital in ADC synthesis. SPDP-sulfo joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T39880	Propargyl-Tos
	Propargyl-Tos is a cleavable linker vital in ADC synthesis. Propargyl-Tos joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T17835	DMAC-PDB	Others	Others
	DMAC-PDB is a cleavable linker vital in ADC synthesis. DMAC-PDB joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T40761	NO2-SPP-sulfo NO2-SPP-sulfo
	NO2-SPP-sulfo is a cleavable linker vital in ADC synthesis. NO2-SPP-sulfo joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T18503	NHS-SS-biotin	Others	Others
	NHS-SS-biotin is a cleavable linker vital in ADC synthesis. NHS-SS-biotin joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T14516	BDP FL DBCO	Others	Others
	BDP FL DBCO is a cleavable linker vital in ADC synthesis. BDP FL DBCO joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T40765	DMAC-SPDB-sulfo
	DMAC-SPDB-sulfo is a cleavable linker vital in ADC synthesis. DMAC-SPDB-sulfo joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T40726	Azide-C2-Azide Azide-C2-Azide
	Azide-C2-Azide is a cleavable linker vital in ADC synthesis. Azide-C2-Azide joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T17539	BCN-SS-amine	Others	Others
	BCN-SS-amine is a cleavable linker vital in ADC synthesis. BCN-SS-amine joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T39023	Biotin-sar-oh
	Biotin-sar-oh is a cleavable linker vital in ADC synthesis. Biotin-sar-oh joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T39087	MC-VC-PAB-NH2 MC-VC-PAB-NH2
	MC-VC-PAB-NH2 is a cleavable linker vital in ADC synthesis. MC-VC-PAB-NH2 joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T40763	NO2-SPDMV-sulfo NO2-SPDMV-sulfo
	NO2-SPDMV-sulfo is a cleavable linker vital in ADC synthesis. NO2-SPDMV-sulfo joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
TP1498	FFAGLDD TFA
	FFAGLDD TFA is an MMP9 selective cleavage peptide, which is used for the cytoplasmic transfer of doxorubicin (DOX) to realize the controlled slow drug delivery and release.
T63434	Abiraterone decanoate
	Abiraterone decanoate 是 Abiraterone 的前药，能够利用肌肉内 (IM) 递送提供 Abiraterone 的受控释放和长效 CYP17 抑制。
T17386	Alkyne-PEG4-SS-PEG4-alkyne	Others	Others
	Alkyne-PEG4-SS-PEG4-alkyne is an eight-unit polyethylene glycol (PEG) linker, designed for antibody-drug conjugates (ADCs) synthesis, that can be cleaved. This linker serves as a connection between the antibody and the drug, allowing for controlled release upon specific conditions [1].
TP1545	FFAGLDD	Others	Others
	FFAGLDD 是 MMP9 选择性切割肽，用于多柔比星 (DOX) 的胞浆递送，实现时间和空间控制的缓慢药物递送和释放。
T18350	Methyltetrazine-PEG4-oxyamine	Others	Others
	Methyltetrazine-PEG4-oxyamine is a 4-unit polyethylene glycol (PEG) linker employed in the synthesis of antibody-drug conjugates (ADCs), which are extensively used for targeted drug delivery [1]. This cleavable linker offers a means to efficiently attach drugs to antibodies and facilitate their controlled release at the target site.
T18521	PC DBCO-PEG3-biotin	Others	Others
	PC DBCO-PEG3-biotin is a trimeric polyethylene glycol (PEG) linker, specifically designed for antibody-drug conjugate (ADC) synthesis, with a cleavable moiety consisting of a dibenzocyclooctyne (DBCO) group and a biotin molecule. This linker provides a platform for the efficient attachment of drugs to antibodies, facilitating the targeted delivery and controlled release of therapeutic agents in ADCs[1].
T18522	PC Mal-NHS carbonate ester	Others	Others
	PC Mal-NHS carbonate ester is a cleavable linker specifically designed for the synthesis of antibody-drug conjugates (ADCs)[1]. This chemical compound plays a crucial role in facilitating the conjugation of drugs to antibodies, enabling targeted delivery and enhanced efficacy of therapeutic agents. Its unique carbonate ester structure allows for efficient cleavage in the targeted environment, ensuring the controlled release of the drug payload. Its application in ADC synthesis highlights its imp...
T38503	(2-pyridyldithio)-PEG1-hydrazine (2-pyridyldithio)-PEG1-hydrazine
	(2-Pyridyldithio)-PEG1-hydrazine is a one-unit cleavable polyethylene glycol (PEG) linker specifically designed for the synthesis of antibody-drug conjugates (ADCs). This linker offers the advantage of controlled release of the drug payload from the ADC construct. It is utilized in the conjugation process between the antibody and the cytotoxic drug, enabling the targeted delivery of the drug to cancer cells. The (2-pyridyldithio) group of this linker provides stability during circulation in the ...
T74437	β-Glucuronide-dPBD-PEG5-NH2
	β-Glucuronide-dPBD-PEG5-NH2 是由 β-葡糖苷酸与 pyrrolobenzodiazepine 通过二聚体形成方式连接，并能与异戊二烯化抗体结合形成抗体-活性分子偶联物 (ADC) cIRCR201-dPBD 的化合物。其所含β-葡糖苷酸键为一种可降解 (cleavable) 的 ADC Linker，作为 cIRCR201-dPBD 的前体能有效减少副作用。此外，β-Glucuronide-dPBD-PEG5-NH2 还具备诱导细胞凋亡 (apoptosis) 和阻滞细胞周期的能力，显示出抗肿瘤活性。
T83742	SBP1 TFA Spike Binding Peptide 1
	Spike binding peptide 1 (SBP1) 为对应于血管紧张素转换酶2 (ACE2) 的第21至43位氨基酸的肽。已将脂质纳米粒子 (LNPs) 包裹的抗病毒化合物奥司他韦磷酸盐与SBP1结合并通过体外研究评估其控制释放奥司他韦磷酸盐的长期潜力。SBP1 (2%) 固定于交联的羟基丙烯酸酯和乙基黄原酸乙酯网络，提高了对严重急性呼吸系统冠状病毒2(SARS-CoV-2)刺突糖蛋白，亦称表面糖蛋白，的网络捕获效率。

化合物

FFAGLDD amine salt

Cat.No: TP1545L1

Target: Others

Fmoc-Ala-Ala-Asn(Trt)-OH

Cat.No: T17946

Target: Others

Diroximel fumarate

Cat.No: T4271

Synonym: Diroximel Fumarete

Target: Others

Cat.No: T14724

Target: Others

Cat.No: T40762

Synonym: NO2-SPDB-sulfo

Cat.No: T18786

Target: Others

Cat.No: T17812

Target: Others

Cat.No: T17836

Target: Others

Cat.No: T18559

Synonym: 2,5-Dioxopyrrolidin-1-yl 3-(pyridin-2-yldisulfanyl)butanoate

Target: Others

Cat.No: T17540

Target: Others

Cat.No: T15927

Target: Others

Cat.No: T39538

Synonym: BCOT-PEF3-OPFP

Azidoethyl-SS-propionic acid

Cat.No: T17524

Target: Others

Tetrazine-biotin

Cat.No: T39169

Cat.No: T40764

Cat.No: T18732

Target: Others

Cat.No: T18505

Target: Others

Cat.No: T38597

Cat.No: T39880

Cat.No: T17835

Target: Others

Cat.No: T40761

Synonym: NO2-SPP-sulfo

Cat.No: T18503

Target: Others

Cat.No: T14516

Target: Others

DMAC-SPDB-sulfo

Cat.No: T40765

Cat.No: T40726

Synonym: Azide-C2-Azide

Cat.No: T17539

Target: Others

Cat.No: T39023

Cat.No: T39087

Synonym: MC-VC-PAB-NH2

NO2-SPDMV-sulfo

Cat.No: T40763

Synonym: NO2-SPDMV-sulfo

Cat.No: TP1498

Abiraterone decanoate

Cat.No: T63434

Alkyne-PEG4-SS-PEG4-alkyne

Cat.No: T17386

Target: Others

Cat.No: TP1545

Target: Others

Methyltetrazine-PEG4-oxyamine

Cat.No: T18350

Target: Others

PC DBCO-PEG3-biotin

Cat.No: T18521

Target: Others

PC Mal-NHS carbonate ester

Cat.No: T18522

Target: Others

(2-pyridyldithio)-PEG1-hydrazine

Cat.No: T38503

Synonym: (2-pyridyldithio)-PEG1-hydrazine

β-Glucuronide-dPBD-PEG5-NH2

Cat.No: T74437

Cat.No: T83742

Synonym: Spike Binding Peptide 1

Cat. No.	Product Name	Target	Signaling Pathways
TN1213	2-(Hydroxymethyl)anthraquinone	Anti-infection	Microbiology/Virology
	2-(Hydroxymethyl)anthraquinone 是光可清除保护基团，在结构上可以阻碍性信息素释放。
T82148	Hydrogenated soya phosphatidylcholines
	Hydrogenated soya phosphatidylcholines 是一种用于提升水溶性药物口服给药效果的天然产物，它能够增加药物负荷和溶解度，从而延长药物释放时间。

天然产物

2-(Hydroxymethyl)anthraquinone

Cat.No: TN1213

Target: Anti-infection

Hydrogenated soya phosphatidylcholines

Cat.No: T82148

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