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Cat. No. Product Name Target Signaling Pathways
T38476 Metallo β-lactamase ligand 1

Antibacterial Microbiology/Virology
Metallo β-lactamase ligand 1 是B 类β-内酰胺酶的抑制剂,具有抗菌活性。
T19206 β-Lactamase-IN-1

4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1

Antibacterial Microbiology/Virology
β-Lactamase-IN-1 (4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one) 是一种 β-Lactamase 抑制剂,针对淋病奈瑟菌的感染。
T35427 β-Lactamase-IN-2

Antibacterial Microbiology/Virology
β-Lactamase-IN-2 是 β-内酰胺酶的有效抑制剂。β-Lactamase-IN-2显示出抗菌活性。
T14979 Clavulanate lithium

Clavulanic acid lithium,克拉维酸锂

Antibacterial Microbiology/Virology
Clavulanate lithium (Clavulanic acid lithium) 是一种β-lactamase 的高效抑制剂,可作抗生素。
T38955 β-Lactamase-IN-4

β-Lactamase-IN-4 (WO2013149121A1, compound 708) is a potent β-lactamase inhibitor. It serves as a valuable tool in the investigation of bacterial infections.
T38956 β-Lactamase-IN-5

β-Lactamase-IN-5, a β-lactamase inhibitor isolated from compound 720, holds significant potential for studying bacterial infections.
T39865 β-Lactamase-IN-6

β-Lactamase-IN-6 is a β-Lactamase inhibitor that shows high antibacetrial activity.
T1631 Sulbactam

CP45899,舒巴坦,舒巴坦酸

Antibacterial; Antibiotic Microbiology/Virology
Sulbactam (CP45899) 是一种竞争性、不可逆的 β-内酰胺酶抑制剂,抑制耐多药不动杆菌-鲍曼不动杆菌复合物。它具有抗菌活性。
T15047 Dacisteine

N,S-Diacetyl-L-cysteine,达西司坦

Others Others
Dacisteine (N,S-Diacetyl-L-cysteine) 是 New Delhi metallo-beta-lactamase-1 (NDM-1) 的抑制剂 (IC50 = 1000 μM)。
T0234 Methicillin sodium salt

Methicillin sodium,Meticillin sodium,甲氧西林钠

Antibacterial; Antibiotic Microbiology/Virology
Methicillin sodium salt 是β-内酰胺抗生素,抑制参与肽聚糖合成的青霉素结合蛋白。
T1143 Carbenicillin disodium

BRL-2064,羧苄青霉素钠,Sodium carbenicillin

Cell wall; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Carbenicillin disodium (BRL-2064) 作用于细菌细胞壁合成的最后阶段,是β-内酰胺青霉素衍生物。
T5570 Cephalothin

头孢噻吩,Cephalotin acid

Antibacterial; Antibiotic Microbiology/Virology
Cephalothin 是一种 β-内酰胺抗生素,抑制 C 类 β-内酰胺酶活性的 Ki 值为 0.32 µM。
T1031 Cloxacillin sodium monohydrate

Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物

Antibacterial; Antibiotic Microbiology/Virology
Cloxacillin sodium monohydrate (Cloxacillin Sodium) 有抗菌作用,对Staphylococcus aureus25923 的最小抑菌浓度为256 mg/L。
T6268 Ceftiofur hydrochloride

头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur hydrochloride (U-67279A) 是头孢噻呋的盐酸盐形式,是一种β-内酰胺酶稳定的半合成广谱头孢菌素,具有抗菌活性。
T0868 Cefepime Dihydrochloride Monohydrate

Cefepime HCl,头孢吡肟二盐酸盐一水合物

Antibacterial; Antibiotic; Antifection Microbiology/Virology
Cefepime Dihydrochloride Monohydrate (Cefepime HCl) 是一种广谱头孢菌素,对革兰氏阳性菌和革兰氏阴性菌有更高的覆盖率。
T1405 Cefditoren pivoxil

头孢妥仑匹酯,ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl

Antibacterial; Antibiotic Microbiology/Virology
Cefditoren pivoxil (ME 1207) 是一种半合成、广谱、β-内酰胺酶耐药的第三代头孢菌素抗生素,具有杀菌活性。
T19860 Clavulanic Acid

BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151

Antibacterial; Antifungal Microbiology/Virology
Clavulanic Acid(RX-10100) 是一种由生物体克拉维链霉菌产生的主要β-内酰胺类抗生素,是一种强效的细菌 β-内酰胺酶抑制剂,用于研究细菌引起的感染。Clavulanic Acid 具有广谱的生物活性,对多种革兰氏阳性和革兰氏阴性细菌均有活性。
T1063 Ticarcillin disodium

Ticarpen,Ticarcillin disodium salt,替卡西林二钠

Antibacterial; Antibiotic Microbiology/Virology
Ticarcillin disodium (Ticarpen) 主要用于抗革兰氏阴性菌, 特别是绿脓杆菌, 也是少数可研究嗜麦芽感染的抗生素。
T1224 Cefuroxime sodium

Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin

Antibacterial; Antibiotic Microbiology/Virology
Cefuroxime sodium (Cefuroxime sodium salt) 是一种具有口服活性的头孢菌素抗生素,增加了对 β-内酰胺酶的稳定性。
T12604 Xeruborbactam

QPX7728

Others Others
QPX7728 is an of ultra-broad-spectrum boronic acid beta-lactamase.
T71613 MK-8712

MK-8712 is a monobactam beta-lactamase inhibitor.
T26906 Brobactam

Brobactam is a beta lactamase inhibitor with antibacterial activity.
T25355 Durlobactam

Durlobactam is a drug candidate for beta-lactamase inhibitor.
T69272 AM-112

AM-112 is an Oxapenem compound which possesses potent beta-lactamase-inhibitory properties.
T75391 Penicillinase

Penicillinase 是一种 β-内酰胺酶。β-内酰胺酶通过水解特征性四元 β-内酰胺环的肽键使抗生素失效,从而使 β-内酰胺抗生素失活。
T69300 AVE-1330A free acid

AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.
T28669 SB 202742

SB202742,SB-202742

SB 202742 is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.
T69299 AVE-1330A sodium

AVE-1330A sodium is a beta-Lactamase inhibitor.
T73438 MK-3402

MK-3402 是一种metallo-beta-lactamase 抑制剂。MK-3402 可用于细菌研究。
T28670 SB 204070 hydrochloride

SB 204070 HCl

SB 204070 hydrochloride is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.
T69999 Nacubactam monohydrate

Nacubactam monohydrate is a beta-lactamase inhibitor used for bacterial infections.
T12524 Potassium clavulanate cellulose

Potassium clavulanate:cellulose (1:1)

Others Others
Potassium clavulanate cellulose is a mixture of potassium clavulanate and cellulose, is an inhibitor of beta-lactamase.
T27386 FR-295389

FR-295389 Free Base,FR295389

FR-295389 is a cephalosporin. FR-295389 shows effective antibacterial activity against metallo-beta-lactamase (MBL)-producers in vitro.
T21163 Cloxacillin Sodium

BRL-1621 sodium salt,Ankerbin,Cloxapen,Austrastaph,BRL 1621 sodium salt

Cloxacillin Sodium, a chlorinated derivative of Oxacillin, is a semi-synthetic antibiotic. Cloxacillin is used for the treatment of infections caused by species of staphylococci which produce beta-lactamase.
T1023 Cefoxitin sodium

Cenomycin,MK-306,头孢西丁钠,Betacef,Merxin

Antibacterial; Antibiotic Microbiology/Virology
Cefoxitin sodium (Betacef) 是一种头霉素类抗生素。Cefoxitin 干扰细胞壁合成。它对革兰氏阴性和革兰氏阳性菌有活性。
T39287 Ledaborbactam

Iedaborbactam, as a beta-lactamase inhibitor (WO2015191907, Example 62), can be used for the research of bacterial infections.
T21384 Dicloxacillin

Dicloxacilina,Dicloxacycline,Dicloxacillinum,Dicloxacilline,Diclocil,Dynapen

Dicloxacillin (INN), a narrow-spectrum β-Lactam antibiotic of the penicillin class, is used against beta-lactamase-producing organisms such as Staphylococcus aureus, which would otherwise be resistant to most penicillins.
T22433 Sulopenem

CP-70429,硫培南

Others Others
Sulopenem, an orally active, potent inhibitor of beta-lactamase, is a parenteral penem antibiotic with broad-spectrum activities against Gram-negative and Gram-positive bacteria.
T1190L Cefmenoxime

A-50912,A 50912,A50912,AB 50912

Cefmenoxime is a cephalosporin antibiotic administered intravenously or intramuscularly. It is an effective inhibitor of Enterobacteriaceae and is resistant to beta-lactamase-initiated hydrolysis. It is active against most common gram-positive and gram-ne
T72261 Metallo-β-lactamase-IN-9

Metallo-β-lactamase-IN-9 (Compound 23) 是一种高效的泛金属-β-内酰胺酶 (MBL) 抑制剂,其对 NDM-1、VIM-1 和 IMP-1 的抑制活性表现在 IC50 值上,分别为 35 nM、269 nM 和 369 nM。
T73668 Sanfetrinem sodium

Sanfetrinem (GV104326) sodium,作为一种β-内酰胺酶稳定的抗生素(antibiotic),对革兰氏阳性菌和革兰氏阴性菌展现出广泛的抗菌活性。
T68938 Cefmenoxime sodium

Cefmenoxime sodium is the ssalt form of Cefmenoxime (free base), a cephalosporin antibiotic administered intravenously or intramuscularly. It is active against most common gram-positive and gram-negative microorganisms. It is a potent inhibitor of Enterobacteriaceae, and is resistant to beta-lactamase-initiated hydrolysis. The drug has a high success rate against many types of infection.
T70621 Cefditoren Pivoxil HCl

Cefditoren Pivoxil is a semi-synthetic, broad-spectrum, beta-lactamase resistant, third-generation cephalosporin antibiotic with bactericidal activity. Cefditoren pivoxil is a prodrug that is rapidly hydrolyzed by intestinal esterases during absorption to the microbiologically active cefditoren, an active aminothiazolyl cephalosporin. Cefditoren inactivates penicillin binding proteins (PBPs) thereby interfering with peptidoglycan synthesis and inhibiting bacterial cell wall synthesis.

化合物

Metallo β-lactamase ligand 1
Cat.No: T38476
Synonym:
Target: Antibacterial
β-Lactamase-IN-1
Cat.No: T19206
Synonym: 4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1
Target: Antibacterial
β-Lactamase-IN-2
Cat.No: T35427
Synonym:
Target: Antibacterial
Clavulanate lithium
Cat.No: T14979
Synonym: Clavulanic acid lithium,克拉维酸锂
Target: Antibacterial
β-Lactamase-IN-4
Cat.No: T38955
Synonym:
Target:
β-Lactamase-IN-5
Cat.No: T38956
Synonym:
Target:
β-Lactamase-IN-6
Cat.No: T39865
Synonym:
Target:
Sulbactam
Cat.No: T1631
Synonym: CP45899,舒巴坦,舒巴坦酸
Target: Antibacterial, Antibiotic
Dacisteine
Cat.No: T15047
Synonym: N,S-Diacetyl-L-cysteine,达西司坦
Target: Others
Methicillin sodium salt
Cat.No: T0234
Synonym: Methicillin sodium,Meticillin sodium,甲氧西林钠
Target: Antibacterial, Antibiotic
Carbenicillin disodium
Cat.No: T1143
Synonym: BRL-2064,羧苄青霉素钠,Sodium carbenicillin
Target: Cell wall, Antibacterial, Antibiotic
Cephalothin
Cat.No: T5570
Synonym: 头孢噻吩,Cephalotin acid
Target: Antibacterial, Antibiotic
Cloxacillin sodium monohydrate
Cat.No: T1031
Synonym: Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物
Target: Antibacterial, Antibiotic
Ceftiofur hydrochloride
Cat.No: T6268
Synonym: 头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride
Target: Antibacterial, Antibiotic
Cefepime Dihydrochloride Monohydrate
Cat.No: T0868
Synonym: Cefepime HCl,头孢吡肟二盐酸盐一水合物
Target: Antibacterial, Antibiotic, Antifection
Cefditoren pivoxil
Cat.No: T1405
Synonym: 头孢妥仑匹酯,ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl
Target: Antibacterial, Antibiotic
Clavulanic Acid
Cat.No: T19860
Synonym: BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151
Target: Antibacterial, Antifungal
Ticarcillin disodium
Cat.No: T1063
Synonym: Ticarpen,Ticarcillin disodium salt,替卡西林二钠
Target: Antibacterial, Antibiotic
Cefuroxime sodium
Cat.No: T1224
Synonym: Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin
Target: Antibacterial, Antibiotic
Xeruborbactam
Cat.No: T12604
Synonym: QPX7728
Target: Others
MK-8712
Cat.No: T71613
Synonym:
Target:
Brobactam
Cat.No: T26906
Synonym:
Target:
Durlobactam
Cat.No: T25355
Synonym:
Target:
AM-112
Cat.No: T69272
Synonym:
Target:
Penicillinase
Cat.No: T75391
Synonym:
Target:
AVE-1330A free acid
Cat.No: T69300
Synonym:
Target:
SB 202742
Cat.No: T28669
Synonym: SB202742,SB-202742
Target:
AVE-1330A sodium
Cat.No: T69299
Synonym:
Target:
MK-3402
Cat.No: T73438
Synonym:
Target:
SB 204070 hydrochloride
Cat.No: T28670
Synonym: SB 204070 HCl
Target:
Nacubactam monohydrate
Cat.No: T69999
Synonym:
Target:
Potassium clavulanate cellulose
Cat.No: T12524
Synonym: Potassium clavulanate:cellulose (1:1)
Target: Others
FR-295389
Cat.No: T27386
Synonym: FR-295389 Free Base,FR295389
Target:
Cloxacillin Sodium
Cat.No: T21163
Synonym: BRL-1621 sodium salt,Ankerbin,Cloxapen,Austrastaph,BRL 1621 sodium salt
Target:
Cefoxitin sodium
Cat.No: T1023
Synonym: Cenomycin,MK-306,头孢西丁钠,Betacef,Merxin
Target: Antibacterial, Antibiotic
Ledaborbactam
Cat.No: T39287
Synonym:
Target:
Dicloxacillin
Cat.No: T21384
Synonym: Dicloxacilina,Dicloxacycline,Dicloxacillinum,Dicloxacilline,Diclocil,Dynapen
Target:
Sulopenem
Cat.No: T22433
Synonym: CP-70429,硫培南
Target: Others
Cefmenoxime
Cat.No: T1190L
Synonym: A-50912,A 50912,A50912,AB 50912
Target:
Metallo-β-lactamase-IN-9
Cat.No: T72261
Synonym:
Target:
Sanfetrinem sodium
Cat.No: T73668
Synonym:
Target:
Cefmenoxime sodium
Cat.No: T68938
Synonym:
Target:
Cefditoren Pivoxil HCl
Cat.No: T70621
Synonym:
Target:
TargetMol Loading
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