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Cat. No. Product Name Target Signaling Pathways
T13554 Arimoclomol maleate

BRX-220

HSP Cytoskeletal Signaling; Metabolism
Arimoclomol maleate (BRX-220) 是一种热休克蛋白 (HSP) 的共诱导剂。它通过增强 Hsp 表达来保护运动神经元,进而通过蛋白酶体-泛素系统直接影响蛋白质聚集和错误折叠装配体的清除
T13553 Arimoclomol

阿瑞洛莫,BRX-220 free base

HSP Cytoskeletal Signaling; Metabolism
Arimoclomol (BRX-220 free base) 是热休克蛋白 (HSP) 的共诱导剂,可用于治疗肌萎缩侧索硬化症的研究。
T40468 Arimoclomol citrate

Arimoclomol citrate,BRX-220 citrate

Arimoclomol citrate (BRX-220 citrate) is a heat shock protein (HSP) co-inducer that acts by enhancing Hsp expression and directly impacting protein aggregation, clearance of misfolded assemblies, and the proteasome-ubiquitin system. This compound is known for its ability to protect motor neurons.
T36470 Biotinyl hexylamine

Biotinyl hexylamine is a synthetic intermediate.1,2It has been used in the synthesis of avidin nucleic acid nano assemblies (ANANAS) and chemotherapeutic conjugates for the diagnosis of, and drug delivery to, tumors. 1.Sabatino, G., Chinol, M., Paganelli, G., et al.A new biotin derivative-DOTA conjugate as a candidate for pretargeted diagnosis and therapy of tumorsJ. Med. Chem.46(14)3170-3173(2003) 2.Bigini, P., Previdi, S., Casarin, E., et al.In vivo fate of avidin-nucleic acid nanoassemblies a...
T37218 N-methyl Mesoporphyrin IX

N-methyl Mesoporphyrin IX 是广泛使用的 G-quadruplex DNA 特异性荧光结合剂,能有效监测 Aβ 纤颤。N-methyl Mesoporphyrin IX 对 G-四链体 DNA 敏感,对双链体、三链体和单链形式的 DNA 没有反应。N-methyl Mesoporphyrin IX 需通过与 Aβ 组装体堆叠才能发出强荧光。同时 N-methyl Mesoporphyrin IX 是一种原位抑制剂,是体外和细胞内 Aβ 淀粉样蛋白生成的非原位监测器。
T82574 DFAME

DFAME为一种帶有红色荧光的基团(Ex=508 nm,Em=641 nm)。它能与二聚体荧光RNA适体Beetroot及Corn结合,分别形成Beetroot-DFAME复合体(Kd=460 nM)和Corn-DFAME复合体(Kd=3600 nM)。这两种复合体可应用于细胞内RNA组装体的形成,利用RNA结构的自组装特性研究RNA纳米结构。

化合物

Arimoclomol maleate
Cat.No: T13554
Synonym: BRX-220
Target: HSP
Arimoclomol
Cat.No: T13553
Synonym: 阿瑞洛莫,BRX-220 free base
Target: HSP
Arimoclomol citrate
Cat.No: T40468
Synonym: Arimoclomol citrate,BRX-220 citrate
Target:
Biotinyl hexylamine
Cat.No: T36470
Synonym:
Target:
N-methyl Mesoporphyrin IX
Cat.No: T37218
Synonym:
Target:
DFAME
Cat.No: T82574
Synonym:
Target:
TargetMol Loading
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