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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T38327 Cryogenine

Cryogenine is an alkaloid originally isolated from H. salicifolia that has anti-inflammatory activity.1 It inhibits prostaglandin synthetase (IC50 = 424 μM). Cryogenine (100 mg/kg per day, p.o.) reduces paw edema and the mean arthritic index in a rat model of adjuvant-induced polyarthritis.2 |1. Lema, W.J., Blankenship, J.W., and Malone, M.H. Prostaglandin synthetase inhibition by alkaloids of Heimia salicifolia. J. Ethnopharmacol. 15(2), 161-167 (1986).|2. Kosersky, D.S., Brown, J.K., and Malon...

化合物

Cryogenine
Cat.No: T38327
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TJS2216 Aurantiamide acetate

金色酰胺醇酯,Asperglaucide

Cysteine Protease Proteases/Proteasome
Aurantiamide acetate (Asperglaucide) 是抑制口服有活性的 cathepsin 选择性抑制剂,分离自 Portulaca oleracea L。它具有抗炎作用,可用于研究炎性相关疾病。

天然产物

Aurantiamide acetate
Cat.No: TJS2216
Synonym: 金色酰胺醇酯,Asperglaucide
Target: Cysteine Protease
TargetMol Loading
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