Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T19763 |
Cetraxate hydrochloride
DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006 |
Serine/threonin kinase | Cell Cycle/Checkpoint; Metabolism |
Cetraxate hydrochloride (DV10062) 是一种有效的顶体蛋白酶 (acrosomal proteinase acrosin) 抑制剂,Ki 和 IC50分别为 0.94 μM 和 3.3 μM。它是一种口服有活性的抗溃疡试剂 (anti-ulcer),具有粘膜保护作用,可用于研究胃溃疡。 | |||
TP1129 |
Boc-Ile-Glu-Gly-Arg-AMC
IEGR-AMC |
||
Boc-Ile-Glu-Gly-Arg-AMC (IEGR-AMC), a specific, highly fluorogenic substrate for clotting enzyme factor Xa (coagulation factor Xa). Boc-IEGR-AMC is also hydrolyzed by acrosin from the ascidian Halocynthia roretzi. |