Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T23543 |
YIL 781
|
GHSR | GPCR/G Protein |
YIL 781是一种选择性ghrelin 受体拮抗剂(GHS-R1a) (Ki = 17 nM)),对运动素受体显示出较弱的亲和力(K = 6 μ M)。YIL 781通过阻断胃饥饿素分泌对体内和体外胰岛素分泌改善体内葡萄糖稳态。 | |||
T29174 |
YIL781 hydrochloride
YIL 781,YIL-781,YIL781 HCl,YIL781 |
||
YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM). |