Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13349 |
WS-383
|
E1/E2/E3 Enzyme | Ubiquitination |
WS-383 是高效、选择性、可逆的DCN1-UBC12相互作用抑制剂,IC50为11 nM。它抑制 Cul3/1 的类泛素化修饰,引起 NRF2,p21和p27 的积累。 | |||
T13348 |
WS-383 free base
|
Others | Others |
WS-383 free base is a selective and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM). |