Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79178 |
WRN inhibitor 2
|
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
WRN inhibitor 2 (example 118)为一WRN(Werner综合征ATP依赖性解旋酶)的抑制剂,其pIC50值不小于7.0。 | |||
T22980 |
MIRA-1
p53 Activator VIII,1-[(1-Oxopropoxy)methyl]-1H-pyrrole-2,5-dione,(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)methyl propionate,NSC 19630,WRN Helicase Inhibitor |
DNA/RNA Synthesis; p53 | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
MIRA-1 (WRN Helicase Inhibitor) 是马来酰亚胺类似物。它可以恢复p53依赖的转录转激活诱导 p53 突变细胞凋亡,具有抗肿瘤作用。 | |||
T72108 | Werner syndrome RecQ helicase-IN-2 | ||
Werner syndrome RecQ helicase-IN-2 (example 57) 是一种有效的 Werner 综合征 RecQ DNA 解旋酶 (WRN) 抑制剂,可用于癌症研究。 |