Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6719 |
Varlitinib
ASLAN001,ARRY-334543 |
HER | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Varlitinib (ASLAN001) 是有效,可逆的泛 EGFR 小分子抑制剂,对 HER1,HER2 和 HER4 的 IC50 值分别为7,2,4 nM。 | |||
T20954 |
Varlitinib Tosylate
Varlitinib-Tosylate,ARRY-334543 Tosylate,ARRY-543 Tosylate |
||
Varlitinib Tosylate is a selective and potent inhibitor of ErbB1(EGFR) and ErbB2(HER2). |