Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0219 |
Valdecoxib
伐地考昔,代他考昔,SC 65872 |
COX | Immunology/Inflammation; Neuroscience |
Valdecoxib (SC 65872) 是可口服的高选择性 COX-2抑制剂,对 COX-2 和 COX-1 的 IC50值分别为 5 nM 和 140 μM,可用于治疗骨关节炎、类风湿性关节炎以及痛经和经期症状。 | |||
T70154 |
1-Hydroxyvaldecoxib
|
||
1-Hydroxyvaldecoxib is a COX-2 inhibitor. | |||
T1780 |
Parecoxib
SC 69124,帕瑞昔布,Vorth-P,Valus-P |
COX | Immunology/Inflammation; Neuroscience |
Parecoxib (SC 69124) 是一种有效的选择性 COX-2 抑制剂,是 Valdecoxib 的前药。 | |||
T1780L |
Parecoxib sodium
SC 69124A,SC-69124A,帕瑞昔布钠,SC69124A,Dynastat |
||
Parecoxib is a cyclooxygenase-2 inhibitor used for the short-term treatment of postoperative pain in adults. Parecoxib is a water-soluble and injectable prodrug of valdecoxib. Parecoxib is a COX2 selective inhibitor in the same category as celecoxib and r |