Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79494 |
VEGFR-2-IN-31
|
VEGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
VEGFR-2-IN-31(compound 3i)是一款针对VEGFR-2的高效抑制剂(IC50=8.93 nM),具有抗前列腺癌的活性。该化合物能够导致细胞周期在S期停滞,并诱导细胞发生凋亡(apoptosis)。 |