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Search Results for " urease "

19

抑制剂 & 化合物

4

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T76107	Urease
	Urease 由多种类型细菌产生，是一些致病菌的有效毒力因子。Urease 还是幽门螺杆菌代谢和毒力的中心，帮助其在胃粘膜中定植。
T67827	Urease Inhibitor 07	Others	Others
	Urease Inhibitor 07 是一种异取代金属蛋白酶抑制剂，对结核分枝杆菌H37Rv 菌株的潜在活性。
T78237	Urease-IN-6
	Urease-IN-6为一种高效Urease抑制剂，IC50值为14.2 μM，适用于消化性溃疡和胃溃疡研究。
T62465	Urease-IN-1
	Urease-IN-1 是一种脲酶抑制剂 (IC50: 2.21±0.45 μM)。
T73047	Urease-IN-5
	Urease-IN-5, 作为一种尿素酶抑制剂，具有1.473 µM的IC50值。该化合物在细胞毒性方面表现较低，并对普通变形杆菌展现出17.78 µg/mL的IC50值的抑制活性。
T64121	Urease-IN-2
	Urease-IN-2 是一种脲酶 (urease) 非竞争性的抑制剂 (IC50: 0.94 μM，Ki: 1.6 μM)，能够非竞争性的抑制 Jack bean 豆脲酶 (JBU)。
T80893	Urease-IN-9
	Urease-IN-9 (Compound 1e) 为脲酶抑制剂，具有IC50值为19.5 μM。
T79656	Urease-IN-8
	Urease-IN-8 (Compound 5e) 为一竞争性脲酶 (Urease) 抑制剂，具IC50值为3.51 μM，Ki值为3.11 μM，主要用于消化性溃疡与胃溃疡研究。
T73046	Urease-IN-4
	Urease-IN-4是一种尿素酶 (urease) 抑制剂，具有1.64 µM的IC50值。此化合物对细胞毒性低，能有效抑制普通变形杆菌，其IC50值为15.27 µg/mL。
T79652	Urease-IN-7
	Urease-IN-7 (Compound 5k)，作为竞争性Urease抑制剂，具有IC50为3.33 μM和Ki值为3.62μM。该化合物可用于消化性溃疡和胃溃疡研究。
T3315	Benurestat 贝奴司他,EU-2826	Others; Antibacterial	Microbiology/Virology; Others
	Benurestat (EU-2826) 是有口服活性的脲酶抑制剂，可研究受感染的尿素分解。
T77348	Butylboronicacid	Others	Others
	Butylboronicacid 是脲酶竞争性抑制剂，可作为单糖络合试剂。
T11305	Flurofamide	Others	Others
	Flurofamide 是一种细菌尿素酶抑制剂，在感染性尿路结石方面有研究的价值。
T1592	Acetohydroxamic acid Methylhydroxamic acid,Acetic acid,Lithostat,AHA,oxime,N-Hydroxyacetamide,乙酰氧肟酸	MMP; Antibacterial	Microbiology/Virology; Proteases/Proteasome
	Acetohydroxamic acid (N-Hydroxyacetamide) 是一种不可逆的细菌和植物尿素酶抑制剂，可研究慢性尿路感染。
T36962	MMP Inhibitor I (trifluoroacetate salt)
	MMP inhibitor I is a peptide inhibitor of matrix metalloproteinase-1 (MMP-1), MMP-2, and MMP-3 (IC50s = 1.3, 30, and 150 μM, respectively). It is selective for MMP-1, MMP-2, and MMP-3 over the proteases thermolysin, urease, trypsin, α-chymotrypsin, plasmin, and elastase at concentrations up to 4 mM.
T78350	Glutamate dehydrogenase
	Glutamate dehydrogenase为存在于原核生物与真核生物线粒体中的酶类，适用于氨、α-酮戊二酸、L-谷氨酸及脲酶的酶促反应检测。
T79450	Enzyme-IN-2
	Enzyme-IN-2（化合物 15），作为ureases抑制剂，展现出了强效的抗尿素分解活性，其Ki值为2.36 μM，而IC50值为0.75 µM。
T36133	3,3'-((2-Chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
	3,3'-((2-Chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one) is a non-nucleotide inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1; Ki = 50 μM).1,2 It also inhibits urease (IC50 = 84.53 μM for the Jack bean enzyme).3 \|1. Choudhary, M.I., Fatima, N., Khan, K.M., et al. New biscoumarin derivatives-cytotoxicity and enzyme inhibitory activities. Bioorg. Med. Chem. 14(23), 8066-8072 (2006).\|2. Onyedibe, K.I., Wang, M., and Sintim, H.O. ENPP1, an old enzyme with new functions, ...
T37832	CAY10761 CAY10761
	CAY10761 is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1; IC50s = 467 and 429 μM for the human and snake venom enzymes, respectively).1,2 It also inhibits mushroom tyrosinase (Ki = 1.9 μM) and urease from jack bean, P. mirabilis, and B. pasteurii (IC50s = 0.093, <0.125, and 0.089 mM, respectively, at pH 8.2).3,4 \|1. Khan, K.M., Fatima, N., Rasheed, M., et al. 1,3,4-Oxadiazole-2(3H)-thione and its analogues: A new class of non-competitive nucleotide pyrophosphatases/p...

化合物

Cat.No: T76107

Urease Inhibitor 07

Cat.No: T67827

Target: Others

Cat.No: T78237

Cat.No: T62465

Cat.No: T73047

Cat.No: T64121

Cat.No: T80893

Cat.No: T79656

Cat.No: T73046

Cat.No: T79652

Cat.No: T3315

Synonym: 贝奴司他,EU-2826

Target: Others, Antibacterial

Butylboronicacid

Cat.No: T77348

Target: Others

Cat.No: T11305

Target: Others

Acetohydroxamic acid

Cat.No: T1592

Synonym: Methylhydroxamic acid,Acetic acid,Lithostat,AHA,oxime,N-Hydroxyacetamide,乙酰氧肟酸

Target: MMP, Antibacterial

MMP Inhibitor I (trifluoroacetate salt)

Cat.No: T36962

Glutamate dehydrogenase

Cat.No: T78350

Cat.No: T79450

3,3'-((2-Chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)

Cat.No: T36133

Cat.No: T37832

Synonym: CAY10761

Cat. No.	Product Name	Target	Signaling Pathways
T4S0578	Guaijaverin 番石榴苷,Guajaverin,Quercetin-3-Arabinoside	Others; Antioxidant; Antibacterial	Microbiology/Virology; Others; oxidation-reduction
	Guaijaverin (Quercetin-3-Arabinoside) 是一种尿素酶抑制剂，IC50值为 120 μM，有抗氧化和抗变形链球菌作用。
TN6604	4-Chlorocinnamic acid
	4-Chlorocinnamic acid is a photosensitive compound. 2-Chlorocinnamic acid and 4-chlorocinnamic acid show potent urease inhibitory activities with the respective IC50 values of 0.66 and 1.10 uM.
TN3465	Atalantoflavone	Antifection	Microbiology/Virology
	Atalantoflavone shows urease inhibitory potential. It displays weak cytotoxic activity against the human Caucasian prostate adenocarcinoma cell line PC-3.
TN6659	2-Chlorocinnamic acid
	2-Chlorocinnamic acid is a photosensitive compound, it can inhibit tyrosinase activity. 2-Chlorocinnamic acid and 4-chlorocinnamic acid show potent urease inhibitory activities with the respective IC50 values of 0.66 and 1.10 uM.

天然产物

Cat.No: T4S0578

Synonym: 番石榴苷,Guajaverin,Quercetin-3-Arabinoside

Target: Others, Antioxidant, Antibacterial

4-Chlorocinnamic acid

Cat.No: TN6604

Atalantoflavone

Cat.No: TN3465

Target: Antifection

2-Chlorocinnamic acid

Cat.No: TN6659

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