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抑制剂 & 化合物

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重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T74662 UBA5-IN-1

UBA5-IN-1 (compound 8.5) 是 UBA5的选择性抑制剂,IC50值为 4.0 μM。UBA5-IN-1 抑制高表达 UBA5 的 Sk-Luci6 癌细胞的增殖。
T7415 DKM 2-93

E1/E2/E3 Enzyme Ubiquitination
DKM 2-93是相对选择性 UBA5抑制剂,IC50=430 μM。

化合物

UBA5-IN-1
Cat.No: T74662
Synonym:
Target:
DKM 2-93
Cat.No: T7415
Synonym:
Target: E1/E2/E3 Enzyme
Cat. No. Product Name Species Expression System
TMPJ-01324 UBA5 Protein, Human, Recombinant (His)

Ubiquitin-like modifier-activating enzyme 5,UBE1DC1...

Human E. coli
UBA5 is a member of the ubiquitin-activating E1 family and UBA5 subfamily. Ubiquitin and ubiquitin-like proteins are recognized as covalently conjugated to various cellular substrates by a three-step enzymatic pathway. The ubiquitin-activating enzyme (E1) has a vital role in the first step of ubiquitination pathway to activate ubiquitin or ubiquitin-like proteins. UBA5 activates ubiquitin-fold modifier 1, a ubiquitin-like post-translational modifier protein, via the formation of a high-energy th...

重组蛋白

UBA5 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01324
Species: Human
Expression System: E. coli
TargetMol Loading
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