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Cat. No. Product Name Target Signaling Pathways
T8520 Tetrazole

1H-TETRAZOLE,1H-四唑

Antibacterial Microbiology/Virology
Tetrazole (1H-TETRAZOLE) 是羧酸的生物等排体,具有相当的抗菌性能。
T6716 Valsartan

Diovan,缬沙坦,Tareg,CGP 48933

RAAS Endocrinology/Hormones
Valsartan (CGP 48933) 是一种血管紧张素 II 受体拮抗剂,有用于高血压和心力衰竭的研究潜力。
T63376 CB 168

CB 168是有效的靶向异亮基 tRNA 合成酶 (IleRS) 选择性氨基酰基氨基酰芳基四唑抑制剂。
T74273 Antifungal agent 52

Antifungal agent 52 (compound 6c) 是四唑衍生物。Antifungal agent 52 抑制麦角固醇 的合成。Antifungal agent 52 对白色念珠菌表现出显着的抗真菌活性 Antifungal agent 52 影响白色念珠菌基底细胞膜通透性。
T78773 Tubulin inhibitor 38

Tubulin inhibitor 38(化合物14)是一款强效的四唑基微管蛋白抑制剂,能够显著抑制细胞增殖。以100 nM浓度作用24小时后,该抑制剂能够引起有丝分裂停滞,特别是在G2/M期细胞周期阶段,进而诱导细胞凋亡。在HeLa、MCF7和U87 MG细胞系中,Tubulin inhibitor 38展现了较高的细胞毒性及选择性。
T38844 MK-8245 Trifluoroacetate

MK-8245 trifluoroacetate is a liver-targeting inhibitor of stearoyl-CoA desaturase (SCD) with IC50 of 1 nM for human SCD1 and 3 nM for both rat SCD1 and mouse SCD1, with anti-diabetic and anti-dyslipidemic efficacy. IC50 value: 1 nM (hSCD1) Target: SCD1 in vitro: MK-8245, a phenoxy piperidine isoxazole derivative, has been identified as a potent and liver-specific SCD inhibitor. It contains a tetrazole acetic acid moiety, which is the key molecule for OATPs recognition and liver-targeting. MK...

化合物

Tetrazole
Cat.No: T8520
Synonym: 1H-TETRAZOLE,1H-四唑
Target: Antibacterial
Valsartan
Cat.No: T6716
Synonym: Diovan,缬沙坦,Tareg,CGP 48933
Target: RAAS
CB 168
Cat.No: T63376
Synonym:
Target:
Antifungal agent 52
Cat.No: T74273
Synonym:
Target:
Tubulin inhibitor 38
Cat.No: T78773
Synonym:
Target:
MK-8245 Trifluoroacetate
Cat.No: T38844
Synonym:
Target:
TargetMol Loading
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