Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79026 |
Tankyrase-IN-5
|
PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Tankyrase-IN-5(Compound 30f)作为MSC2504877的类似物,能有效抑制tankyaseTNKS1和TNKS2,其IC50分别为2.3 nM和7.9 nM。 |