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Cat. No. Product Name Target Signaling Pathways
T13212 TRPA1 Antagonist 1

TRP/TRPV Channel Membrane transporter/Ion channel
TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.
T40822 TRPA1 Antagonist 3

TRPA1 Antagonist 3

TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.
T64337 PF-04745637

PF4745637,PF 4745637,PF 04745637,PF-4745637

TRP/TRPV Channel Membrane transporter/Ion channel
PF-04745637 是TRPA1的选择性拮抗剂,对人 TRPA1 的IC50为 17 nM。
T25078 AMG9090

AMG 9090,AMG-9090

AMG9090 is a transient receptor potential ankyrin 1 (TRPA1) antagonist.
T39935 TRPA1-IN-1

TRPA1-IN-1

TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.

化合物

TRPA1 Antagonist 1
Cat.No: T13212
Synonym:
Target: TRP/TRPV Channel
TRPA1 Antagonist 3
Cat.No: T40822
Synonym: TRPA1 Antagonist 3
Target:
PF-04745637
Cat.No: T64337
Synonym: PF4745637,PF 4745637,PF 04745637,PF-4745637
Target: TRP/TRPV Channel
AMG9090
Cat.No: T25078
Synonym: AMG 9090,AMG-9090
Target:
TRPA1-IN-1
Cat.No: T39935
Synonym: TRPA1-IN-1
Target:
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