Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1997L |
[Ala17]-MCH acetate
[Ala17]-MCH acetate(359784-84-2 free base) |
Melanin-concentrating Hormone Receptor (MCHR) | GPCR/G Protein |
[Ala17]-MCH acetate 是 MCHR1 的选择性配体,Ki 为 0.16 nM,Kd 为 0.37 nM(Eu3+ 螯合物标记)。 [Ala17]-MCH acetate 对 MCHR2 具有选择性,Ki 为 34 nM。 | |||
TP1997 |
[Ala17]-MCH
|
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Potent melanin-concentrating hormone (MCH) receptor agonist (EC50 values are 17 and 54 nM at MCH1 and MCH2 receptors respectively). Displays some selectivity towards MCH1 over MCH2 (Ki values are 0.16 and 34 nM respectively). |