Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8485 |
THIQ
|
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
THIQ 是一种选择性黑皮质素 4 受体 (MC4R) 激动剂,对 hMC4R 和 rMC4R 的 IC50 分别为 1.2 和 0.6 nM。 | |||
T34858 |
THIQ-20c
THIQ 20c |
||
THIQ-20c is a steroidomimetic and chimeric microtubule disruptor. | |||
T70179 |
THIQ-40
|
||
THIQ-40 is a novel potent erα antagonist and selective estrogen receptor degrader (serd), exhibiting good oral bioavailability, antitumor efficacy, and serd activity in vivo | |||
T70178 |
Sonidegib metabolite M25
|
||
Sonidegib metabolite M25 is a smoothened (SMO) antagonist. |