Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4965L |
TCS-OX2-29 HCl
TCSOX 229,TCS-OX229,TCS OX229,TCS OX2 29,TCSOX-229,TCSOX229 |
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TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation. | |||
T4965 |
TCS-OX2-29
|
OX Receptor | GPCR/G Protein; Neuroscience |
TCS-OX2-29 是高亲和力和选择性OX2R 拮抗剂,IC50值为 40 nM,pKI 值为 7.5。它对 OX2 的选择性比 OX1 高 250 倍以上。 |