Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T68213 |
Palonidipine HCl
|
||
Palonidipine HCl is a calcium channel antagonist potentially for the treatment of angina pectoris and hypertension. | |||
T17009 |
TC-S 7009
|
HIF | Angiogenesis; Chromatin/Epigenetic |
TC-S 7009是一种有效的和具有选择性的HIF-2α抑制剂(Kd: 81 nM)。TC-S 7009对HIF-2α的亲和力大于HIF-1α (Kd >> 5 μM)。 TC-S 7009破坏HIF-2α异源二聚化,降低HIF-2α靶基因表达,降低dna 结合活性。 |