Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T23458 |
THZ1 Hydrochloride (1604810-83-4 free base)
THZ1 Hydrochloride |
Others | Others |
THZ1 is a covalent inhibitor of CDK7 (IC50: 3.2nM). | |||
T13153 |
THZ1-R
|
CDK | Cell Cycle/Checkpoint |
THZ1-R displays diminished activity for CDK7 inhibition(Kd:142 nM). | |||
T3664 |
THZ1
CDK7 inhibitor,THZ1 2HCl |
CDK | Cell Cycle/Checkpoint |
THZ1 (CDK7 inhibitor) 是一种新型的选择性强效共价 CDK7 抑制剂。它还抑制CDK12和CDK13,并下调 MYC 表达。 | |||
T72512 |
THZ1 Hydrochloride
|
||
THZ1 Hydrochloride,一种有效、选择性的共价CDK7抑制剂,IC50值为3.2 nM。它同样针对相关激酶CDK12和CDK13具有抑制作用,并能下调MYC表达。 |