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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T36844 Inostamycin A

Inostamycin A is a bacterial metabolite that has been found inStreptomycesand has anticancer activity.1It is an inhibitor of CDP-diacylglycerol:inositol 3-phosphatidyltransferase (IC50= 0.02 μg/ml in A431 cell membranes) and is selective for CDP-diacylglycerol:inositol 3-phosphatidyltransferase over phospholipase C (PLC) and phosphatidylinositol kinase at 10 μg/ml.2Inostamycin A decreases viability of YCU-T892, KCC-TC873, KB, HSC-4, and YCU-T891 oral squamous cell carcinoma (OSCC) cells in a con...

化合物

Inostamycin A
Cat.No: T36844
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1678 Nystatin

Stamycin,Fungicidin,制霉菌素,Nystavescent

Apoptosis; Antibiotic; Antifungal Apoptosis; Microbiology/Virology
Nystatin (Fungicidin) 是一种口服对酵母和支原体有效的多烯类抗真菌抗生素。它能增加质膜对包括氯离子等小单价离子的通透性。它可部分阻止 Oxaliplatin 诱导的脂筏聚集、DR4 和 DR5 聚集的胆固醇隔离试剂,减少细胞凋亡。
T1214 Ribostamycin sulfate

Vistamycin sulfate,硫酸核糖霉素

Antibacterial; Antibiotic Microbiology/Virology
Ribostamycin sulfate (Vistamycin sulfate) 是一种广谱抗菌剂, 在30S 和50S 核糖体亚基结合抑制细菌蛋白质合成, 还抑制蛋白二硫键异构酶分子伴侣活性, 用于药代动力学和肾毒性研究。
T73730 Distamycin A

Distamycin A (NSC-82150)为一种寡肽抗生素及小沟结合剂,其结合B型DNA,并倾向于A/T富集区。Distamycin A能调节烯二炔诱导DNA切割位点并促进细胞凋亡。
T74207 Ribostamycin

Ribostamycin (Vistamycin) 是一种广谱氨基糖苷类抗生素 (antibiotic)。Ribostamycin 对革兰氏阴性和革兰氏阳性细菌感染有效。Ribostamycin 还抑制PDI 的伴侣活性。

天然产物

Nystatin
Cat.No: T1678
Synonym: Stamycin,Fungicidin,制霉菌素,Nystavescent
Target: Apoptosis, Antibiotic, Antifungal
Ribostamycin sulfate
Cat.No: T1214
Synonym: Vistamycin sulfate,硫酸核糖霉素
Target: Antibacterial, Antibiotic
Distamycin A
Cat.No: T73730
Synonym:
Target:
Ribostamycin
Cat.No: T74207
Synonym:
Target:
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