Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9446 |
KB-0742 dihydrochloride
|
CDK | Cell Cycle/Checkpoint |
KB-0742 dihydrochloride 是一种有效的、选择性的、口服的 CDK9 抑制剂,具有抗肿瘤活性,对CDK9/cyclin T1的IC50为 6 nM。它对CDK9/cyclin T1具有选择性,其选择性是其他 CDK 激酶的 50 倍以上。 | |||
TP1641 |
[pSer2, pSer5, pSer7]-CTD TFA
|
||
[pSer2, pSer5, pSer7]-CTD (TFA) is a substrate for CDK7(cyclin-dependent protein kinase), a phosphorylated polypeptide at ser2, ser5, and ser7 of RNA polymerase II carboxyl terminus (CTD). | |||
TP1683 |
[pSer2, pSer5, pSer7]-CTD
|
||
[pSer2, pSer5, pSer7]-CTD is a substrate for CDK7(cyclin-dependent protein kinase), a phosphorylated polypeptide at ser2, ser5, and ser7 of RNA polymerase II carboxyl terminus (CTD). |