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Cat. No. Product Name Target Signaling Pathways
T12930 SKF89976A hydrochloride

d,l-SKF89976A hydrochloride

GABA Receptor Membrane transporter/Ion channel; Neuroscience
SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) 是GABA 转运蛋白GAT-1的选择性抑制剂,抑制 CHO 细胞中的 GAT-1,GAT-2 和 GAT-3,IC50分别为 0.28 μM,137.34 μM 和 202.8 μM。
T68550 SKF89976A HCl

SKF89976A is a potent GABA uptake inhibitor, which is selective for GAT-1 (IC50 values are 0.13, 550, 944 and 7210 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively). SKF89976A inhibits transport current competitively (Ki = 7 μM) and transmitter-gated current non-competitively (Ki = 0.03 nM). It is able to pass the blood-brain barrier after systemic administration and is active in vivo.

化合物

SKF89976A hydrochloride
Cat.No: T12930
Synonym: d,l-SKF89976A hydrochloride
Target: GABA Receptor
SKF89976A HCl
Cat.No: T68550
Synonym:
Target:
TargetMol Loading
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