Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2255 |
SB-743921 hydrochloride
SB743921 HCl,SB743921 |
Kinesin; KSP | Cell Cycle/Checkpoint; Cytoskeletal Signaling |
SB-743921 hydrochloride (SB743921 HCl) 是一种有效的驱动蛋白纺锤体蛋白 KSP 抑制剂,Ki 值为 0.1 nM。 | |||
T28694 |
SB-743921 free base
SB743921,SB-921,SB921,SB-743921,GSK-743921,GSK-921 |
||
SB-743921, a kinesin spindle protein (KSP) inhibitor, is used potentially for the treatment of non-Hodgkin's lymphoma (NHL). | |||
T81871 | Mal-PEG8-Val-Ala-PAB-SB-743921 | ||
Mal-PEG8-Val-Ala-PAB-SB-743921 (Compound D7) 是一种用于 ADC 的药物-Linker偶联物。由KSP抑制剂SB-743921和连接子组成,此合成物可应用于ADC合成过程。 |