Cat. No. | Product Name | Target | Signaling Pathways |
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T72446 |
SARS-CoV-2 Mpro-IN-4
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SARS-CoV-2 Mpro-IN-4是针对主要蛋白酶(MPro)和组织蛋白酶L(CatL)的双重抑制剂,其IC50s分别为900 nM和60 nM。此化合物对SARS-CoV2展现出抗病毒活性,在hACE2表达的A549细胞中可有效阻断SARS-CoV2复制,其IC50值为8.2 nM。 | |||
T38175 |
MPro N3
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Coronavirus main protease (Mpro) inhibitor (respective IC50 values are 2.7, 4 and 8.8 μM for MHV-A29, HCoV-229E and FOPV replication in vitro). Inhibits viral cell infection in an MHV plaque reduction assay. Also inhibits SARS-CoV-2 viral cell entry in a plaque reduction assay (IC50 = 16.8 μM). |