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Cat. No. | Product Name | Target | Signaling Pathways |
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T40340 |
SARS-CoV-2-IN-10
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SARS-CoV-2-IN-10 is a powerful and non-toxic inhibitor of SARS-CoV-2 3CL protease, with IC50 and EC50 values of 0.13 nM and 1.03 nM, respectively. The SARS-CoV-2 3C-like protease (3CLpro) is a critical enzyme for viral replication and serves as an ideal target for intervention. By targeting the SARS-CoV-2 3CL protease, SARS-CoV-2-IN-10 has the potential to facilitate the development of effective antiviral drugs specific to SARS-CoV-2. | |||
T72312 |
SARS-CoV-2 3CLpro-IN-10
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SARS-CoV-2 3CLpro-IN-10(5d)为一种有效的抗 SARS-CoV-2 3CL 蛋白酶抑制剂,其IC50值仅为190 nM,同时对SARS-CoV-1的IC50值为790 nM,对MERS-CoV的IC50值则为70 nM,显示出广谱的抗病毒活性。 | |||
T79515 |
SARS-CoV-2 Mpro-IN-10
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SARS-CoV | Microbiology/Virology |
SARS-CoV-2 Mpro-IN-10(27h)是Mpro抑制剂,具有IC50和EC50值分别为10.9 nM和43.6 nM,适用于SARS-CoV-2病毒的研究。 | |||
T79278 |
SARS-CoV-2 Mpro-IN-7
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SARS-CoV | Microbiology/Virology |
Mpro-IN-7(化合物6g)是一种针对Mpro-SARS-CoV-2的高效抑制剂,具有IC50值为8.8 μM,CC50值为10 μM。 | |||
T62410 |
Hydroxyethylamine
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Hydroxyethylamine (Compd VII) 是一种 SARS-CoV-2 3CLpro 抑制剂,在传播试验中的IC50为 ~10 μM。Hydroxyethylamine 表现出显著的抗病毒效果。 | |||
T37776 | FASN-IN-4 tosylate | ||
FASN-IN-4 tosylate 是高效的脂肪酸合酶 FASN 抑制剂,IC50值为 10 nM。FASN-IN-4 tosylate 还抑制 SARS-CoV-2,EC50为 18.6 nM。 | |||
T78765 |
SARS-CoV-2-IN-51
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SARS-CoV | Microbiology/Virology |
SARS-CoV-2-IN-51(S-10)为针对Omicron的融合抑制剂有效先导化合物,具有抑制Omicron及其他变体的能力,EC50值介于0.82-5.45 μM之间。该化合物通过与SARS-CoV-2病毒S蛋白预融合状态下直接相互作用,从而抑制病毒进入。 | |||
T62829 | SARS-CoV-2 nsp14-IN-1 | ||
SARS-CoV-2 nsp14-IN-1 (Compound 3) 是一种典型的 SARS-CoV-2Nsp14 Mtase 双底物抑制剂 (IC50: 0.061 μM)。SARS-CoV-2 nsp14-IN-1 对人类甲基转移酶表现出良好的选择性,可拮抗 10 种人甲基转移酶(如组蛋白赖氨酸、蛋白精氨酸、DNA 和 RNA 等)。 | |||
T38174 | Mpro inhibitor N3 hemihydrate | ||
Mpro inhibitor N3 hemihydrate is a potent inhibitor of SARS-CoV-2 Mpro with an EC50 of 16.77 μM for SARS-CoV-2. Mpro inhibitor N3 hemihydrate specifically inhibits Mpro from multiple coronaviruses, including SARS-CoV and MERS-CoV. Mpro inhibitor N3 hemihydrate displays inhibition against HCoV-229E, FIPV, and MHV-A59 with individual IC50 of 4.0 μM, 8.8 μM, and 2.7 μM, respectively[1][2]. Mpro inhibitor N3 hemihydrate (0-0.64 μM) is able to penetrate cells to inhibit the replication of IBV viruses... |
Cat. No. | Product Name | Target | Signaling Pathways |
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T79947 |
10-Hydroxyaloin A
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SARS-CoV | Microbiology/Virology |
10-Hydroxyaloin A有效抑制SARS-CoV-2,与SARS-CoV-2 Mpro活性位点显著结合。 |