Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T23283 |
2-Methoxyidazoxan monohydrochloride
RX 821002 hydrochloride |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
L-Albizziin (2-Methoxyidazoxan monohydrochloride) 是高效的 alpha 2r 肾上腺素受体选择性拮抗剂,对 imidazoline 拮抗作用很小或没有。它对 (豚鼠) alpha 2D 肾上腺素受体 (pKd9.7) 的亲和力明显高于 (兔子) alpha 2A 肾上腺素受体 (pKd8.2)。 | |||
T28631 |
RX821002
RX-821002,RX 821002 |
||
RX821002 is a potent and selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. RX821002 displays selectivity for the α2D over the α2A subtypes (pKd values are 9.7 and 8.2 respectively). |