Cat. No. | Product Name | Target | Signaling Pathways |
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T63433 | RSV-IN-5 | ||
RSV-IN-5 是有效的野生型和突变呼吸道合胞病毒 (RSV) 融合蛋白的双重抑制剂。RSV-IN-5 能够作用于野生型 A2 F 蛋白及 D486N 突变 F 蛋白,他们的EC50值分别为2.0 nM、8.1 nM,表现出有效的抗 RSV 作用。 | |||
T79221 |
RSV L-protein-IN-5
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RSV | Microbiology/Virology |
RSVL-protein-IN-5(compound E)是一种高效针对呼吸道合胞病毒(RSV)的抑制剂,拥有EC50值为0.1 μM。该化合物在IC50为0.66 μM的条件下能够抑制聚合酶(Polymerase),并通过阻断病毒转录物的鸟苷酸化过程来抑止RSVmRNA的合成。RSVL-protein-IN-5具有中等细胞毒性(CC50为10.7 μM,HEp-2细胞),同时,在每日4.1 mg/kg剂量下,能减少RSV感染小鼠模型中的病毒滴度。 | |||
T38297 |
Ribavirin-13C5
Ribavirin-13C5 |
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Ribavirin-13C5is intended for use as an internal standard for the quantification of ribavirin by GC- or LC-MS. Ribavirin is an antiviral guanosine nucleoside analog.1,2Upon entry into cells, ribavirin is metabolized to an active triphosphate form that induces viral RNA chain termination and inhibits viral polymerases. It reduces replication in a panel of seven RNA and four DNA viruses in Vero cells (EC50s = 2-95 μg/ml).3Ribavirin also reduces replication of severe acute respiratory syndrome coro... |