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Cat. No. Product Name Target Signaling Pathways
T79518 ROS inducer 3

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
ROS inducer 3 (Compound I6) 是活性氧诱导剂,体外活性良好,其 EC50 值为 2.86 μg/mL。该化合物在体内展现对 Pseudomonas syringae pv. actinidiae 的卓越生物活性,因此可作为研究难治性植物细菌性疾病的杀菌剂。
T36514 QD-394

QD-394 is an inducer of reactive oxygen species (ROS) production.1It induces lipid peroxidation, increases in intracellular accumulation of reactive oxygen species (ROS), and decreases in the reduced glutathione (GSH) to oxidized GSH (GSSG) ratio in MIA PaCa-2 pancreatic cancer cells when used at concentrations ranging from 0.5 to 10 μM. QD-394 is cytotoxic to MIA PaCa-2, PANC-1, and BxPC-3 cancer cells (IC50s = 0.64, 0.34, and 0.9 μM, respectively). QD-394 acts synergistically with napabucasin ...
T79359 Anticancer agent 147

Ferroptosis Apoptosis
Anticanceragent 147(化合物6j),作为槐定碱的衍生物,功能为铁死亡(Ferroptosis)诱导剂。该化合物能促进Fe2+、活性氧(ROS)及丙二醛(MDA)在细胞内的积累,并通过增加内质网(ER)应激和上调转录因子ATF3的表达发挥作用。在体外及体内实验中,Anticanceragent 147展现了出色的抗肝癌活性。

化合物

ROS inducer 3
Cat.No: T79518
Synonym:
Target: Reactive Oxygen Species
QD-394
Cat.No: T36514
Synonym:
Target:
Anticancer agent 147
Cat.No: T79359
Synonym:
Target: Ferroptosis
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