Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6922 |
ORY1001
RG-6016,ORY-1001 (RG-6016) 2HCl,ORY-1001,ORY 1001 |
Histone Demethylase | Chromatin/Epigenetic |
ORY1001 (ORY 1001) 是一种具有口服活性的选择性赖氨酸特异性去甲基化酶 LSD1/KDM1A 抑制剂,对相关的 FAD 依赖性氨氧化酶具有高选择性,IC50 <20 nM。 | |||
T5825 |
Iadademstat dihydrochloride
ORY-1001(trans) |
Histone Demethylase | Chromatin/Epigenetic |
Iadademstat dihydrochloride (ORY-1001(trans)) 是一种不可逆的选择性赖氨酸特异性脱甲基酶 1A(KDM1A/LSD1) 抑制剂,用于治疗急性白血病。 | |||
T28269 |
ORY-1001 free base
RG 6016,ORY-1001,ORY 1001,ORY1001,RG-6016,RG6016 |
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ORY-1001 is a KDM1A inhibitor (IC50 <20nM) with high selectivity against related FAD dependent aminoxidases (MAO-A/B, IL4I1, KDM1B >100uM, SMOX 7uM). Treatment of THP-1 (MLL-AF9) cells with ORY-1001, results in a time/dose dependent me2H3K4 accumulation a |