Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4370 |
Resminostat hydrochloride
4SC-201 hydrochloride,RAS2410 hydrochloride |
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Resminostat hydrochloride (RAS2410 hydrochloride) 是HDAC1,HHDAC3和HDAC6抑制剂,IC50值分别为 42.5、50.1和71.8 nM,对 HDAC8 的活性较低,IC50值为 877 nM。 | |||
T6637 |
Resminostat
马西替坦,4SC-201,RAS2410 |
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Resminostat (4SC-201) 是一种可口服的HDAC1、HDAC3和HDAC6抑制剂,IC50值分别为 42.5、50.1和71.8 nM,具有潜在抗肿瘤活性。 |