Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6336 |
Amonafide
NSC308847,AS1413,氨萘非特,Nafidimide,AS1413,Quinamed |
Topoisomerase | DNA Damage/DNA Repair |
Amonafide (NSC-308847,AS1413) 是一种拓扑异构酶 II 的抑制剂和 DNA 的嵌入剂,通过拓扑异构酶 II 介导的反应产生蛋白质相关的 DNA 链断裂 | |||
T70531 |
CGP 55845
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CGP 55845 is a potent, selective GABAB receptor antagonist (IC50 = 5 nM) that prevents agonist binding (pKi = 8.35) and inhibits GABA and glutamate release (pEC50 values are 8.08 and 7.85 respectively). |