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Cat. No.	Product Name	Target	Signaling Pathways
T20898	(R)-Propranolol hydrochloride Dexpropranolol hydrochloride,(R)-(+)-Propranolol,盐酸普奈洛尔	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) 是一种抗肾上腺素受体拮抗剂，是一种普萘洛尔的活性较低的对映体。Dexpropranolol 是一种非选择性的β-adrenergic receptor 拮抗剂，对 β1AR 和 β2AR 具有高亲和力。
T23302	(S)-(-)-Propranolol hydrochloride	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。
T12550	Propranolol-d7 hydrochloride Propranolol D7 hydrochloride	Others	Others
	Propranolol D7 hydrochloride is a deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective antagonist of β-adrenergic receptor (βAR).
T36237	5-hydroxy Propranolol
	5-hydroxy Propranolol is a metabolite of propranolol , a β-adrenergic receptor antagonist. Propranolol is primarily metabolized in the liver, with cytochrome P450 isoform 2D6 directing ring hydroxylation and the generation of 5-hydroxy propranolol and related metabolites.
T36231	rac-7-hydroxy Propranolol (hydrochloride)
	rac-7-hydroxy Propranolol (hydrochloride) is a ring-hydroxylated isomer and metabolite of propranolol that is an antagonist at β-adrenergic receptors (0.95 potency relative to propranolol). It also demonstrates potent vasodilator activity (0.20 potency relative to propranolol; pA2 = 7.58).
T35402	(±)-4-hydroxy Propranolol β-D-Glucuronide
	(±)-4-hydroxy Propranolol β-D-glucuronide is a metabolite of (±)-4-hydroxy propranolol , which is a metabolite of propranolol. The apparent half-life of (±)-4-hydroxy propranolol β-D-glucuronide is similar to propranolol and 4-hydroxy propranolol. Propranolol is a β-adrenergic antagonist, and the active enantiomer, (S)-(-)-propranolol , has log Kd values of -8.16, -9.08, and -6.93 for β1, β2, and β3, respectively.
T10150	4-Hydroxypropranolol hydrochloride (±)-4-hydroxy Propranolol hydrochloride	Others	Others
	4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors (pA2s: 8.24 and 8.26).
T10149	4-Hydroxypropranolol-d7 hydrochloride (±)-4-hydroxy Propranolol D7 hydrochloride,4-Hydroxypropranolol D7 hydrochloride	Others	Others
	4-Hydroxypropranolol D7 hydrochloride is deuterium-labeled 4-Hydroxypropranolol hydrochloride. 4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors
T78835	Phosphatase-IN-1	Antifungal	Microbiology/Virology
	Phosphatase-IN-1（compound II-8）是Propranolol的衍生物，充当磷脂酸磷酸酶（Pah）的抑制剂。Phosphatase-IN-1能够与 MoPah1结合，展现出19.8 μM的亲和常数。Phosphatase-IN-1能够抑制植物病原体的生长，并显示出抗真菌特性，同时对稻苗和麦穗表现出无毒性。
T34124	Pranolium UM-272,SC-27761,UM 272,SC 27761,SC27761
	Pranolium is a quaternary dimethyl derivative of Propranolol, a well-known powerful betareceptor-blocking agent.
T70506	Bupranolol HCl
	Bupranolol is a non-selective beta blocker without intrinsic sympathomimetic activity (ISA), but with strong membrane stabilizing activity. Its potency is similar to propranolol. Bupranolol is quickly and completely absorbed from the gut. Over 90% undergo first-pass metabolism. Bupranolol has a plasma half life of about two to four hours, with levels never reaching 1 µg/l in therapeutic doses. The main metabolite is carboxybupranolol, 4-chloro-3-[3-(1,1-dimethylethylamino)-2-hydroxy-propyloxy]be...