Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1577 |
Midodrine hydrochloride
Pro-Amatine,盐酸米多君 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Midodrine hydrochloride (Pro-Amatine) 通过去甘氨酸反应转化为其活性代谢物 desglymidodrine。Desglymidodrine 选择性地结合并激活小动脉和静脉血管系统的 α-1-肾上腺素能受体。这会导致平滑肌收缩并导致血压升高。 Desglymidodrine 在血脑屏障中的扩散很差,因此与对中枢神经系统的影响无关。Midodrine hydrochloride 是 midodrine 的盐酸盐形式,是一种直接作用的前药和拟交感神经药,具有抗低血压特性。 | |||
T33384 |
Midodrine (R-isomer HCl)
ProAmatine,Midodrine,ST-1085,Gutron,Amatine |
||
Midodrine is a vasopressor/antihypertensive agent for the treatment of symptomatic postural hypotension. | |||
T22369 |
Midodrine
米多君,(±)-Midodrin |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Midodrine ((±)-Midodrin) 是α1受体激动剂,用于研究家族性自主神经异常以及直立性低血压。 | |||
T12035 |
Midodrine D6 hydrochloride
盐酸米多君 D6 |
Others | Others |
Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent. |