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Cat. No. Product Name Target Signaling Pathways
T75994 SPR741 TFA

SPR741 TFA (NAB741 TFA),一种源自多粘菌素B的阳离子肽增效剂,通过提升革兰氏阴性细菌外膜通透性用于对抗重度革兰氏阴性细菌感染。它能够抑制多重耐药性革兰氏阴性细菌,并在与抗生素联用时扩大抗生素的活性谱。
T35742 IKD-8344

IKD-8344 is a macrocyclic dilactone originally isolated from an actinomycete species and has diverse biological activities, including anticancer, antimicrobial, and anthelmintic properties.1,2,3 It is cytotoxic to L5178Y murine leukemia cells (IC50 = 0.54 ng/ml).1 IKD-8344 inhibits growth of the mycelial form of C. albicans (MIC = 6.25 μg/ml) and potentiates the activity of polymyxin B against the multidrug-resistant pathogenic bacterium B. cenocepacia.2,3 It is active against T. spiralis in vit...

化合物

SPR741 TFA
Cat.No: T75994
Synonym:
Target:
IKD-8344
Cat.No: T35742
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T25971 Polymyxin B2

Polymyxin-B2,PolymyxinB2

Polymyxin B2 is an antibiotic primarily utilized for resistant Gram-negative infections. It is derived from the bacterium Bacillus polymyxa.
T83903 Polymyxin B2 sulfate

Polymyxin B2是一种抗生素,并且是从B. polymyxa分离出的阳离子脂肽抗生素polymyxin B的主要成分。该化合物对P. aeruginosa、A. baumannii、K. pneumoniae和E. cloacae菌株具有活性(MICs分别为1-2、0.5-1、0.25-0.5和0.25-1 µg/ml)。在体内实验中,以4 mg/kg剂量的Polymyxin B2能显著降低P. aeruginosa血液感染小鼠模型中的血液集落形成单位(CFUs)数量。
T83902 Polymyxin E1 sulfate

Colistin A sulfate

Polymyxin E1,是一种肽类抗生素,也是原初从B. polymyxa分离得到的阳离子脂肽抗生素colistin的主要成分。对P. aeruginosa和E. coli具有活性(MICs分别为2和0.8 µg/ml)。

天然产物

Polymyxin B2
Cat.No: T25971
Synonym: Polymyxin-B2,PolymyxinB2
Target:
Polymyxin B2 sulfate
Cat.No: T83903
Synonym:
Target:
Polymyxin E1 sulfate
Cat.No: T83902
Synonym: Colistin A sulfate
Target:
TargetMol Loading
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