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Search Results for " pilocarpine "

4

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T23508 VU 0255035

AChR Neuroscience
VU 0255035 是高度选择性、竞争性和血脑屏障通透性的毒蕈碱 M1 受体拮抗剂,IC50为 130 nM,可减少毛果芸香碱诱导的小鼠癫痫发作。
T13615 Cinperene

桂哌林,R5046

Others Others
Cinperene is an atropine-like compound that can block pilocarpine-induced salivation and lacrimation.
T70292 DDPM-2571 HCl

DDPM-2571 is a highly potent and in vivo active inhibitor of GABA transporter subtype 1 with anticonvulsant, anxiolytic, antidepressant and antinociceptive properties. DDPM-2571 was quickly distributed into the brain and was highly effective in the prevention of chemically-induced seizures (pentylenetetrazole and pilocarpine models) and 6-Hz convulsions. It demonstrated significant anxiolytic-like and antidepressant-like properties. DDPM-2571 had antinociceptive properties, both in the hot plate...
T81674 NIR-FP

NIR-FP是一款用于超氧阴离子(O2-)检测的近红外荧光探针,具备高灵敏度和高选择性。由于O2-是活性氧种(ROS)的关键前体,此探针能有效动态监测由超氧阴离子引发的铁死亡介导的癫痫模型。这些模型包括红藻氨酸诱导的慢性癫痫模型、Pentylenetetrazole诱导的急性癫痫模型以及毛果芸香碱诱导的癫痫模型。

化合物

VU 0255035
Cat.No: T23508
Synonym:
Target: AChR
Cinperene
Cat.No: T13615
Synonym: 桂哌林,R5046
Target: Others
DDPM-2571 HCl
Cat.No: T70292
Synonym:
Target:
NIR-FP
Cat.No: T81674
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0804 Pilocarpine Hydrochloride

NSC 5746 HCl,盐酸毛果芸香碱,Pilocarpine HCl,(+)-Pilocarpine hydrochloride

AChR Neuroscience
Pilocarpine Hydrochloride (NSC 5746 HCl) 是一种 M3 型毒蕈碱乙酰胆碱受体激动剂,用于制作癫痫实验模型
T1231 Pilocarpine nitrate

匹鲁卡品硝酸盐,Pilagan,硝酸毛果芸香碱,Pilofrin

AChR Neuroscience
Pilocarpine nitrate (Pilagan) 是 M3 型毒蕈碱乙酰胆碱受体激动剂,可用于治疗青光眼。

天然产物

Pilocarpine Hydrochloride
Cat.No: T0804
Synonym: NSC 5746 HCl,盐酸毛果芸香碱,Pilocarpine HCl,(+)-Pilocarpine hydrochloride
Target: AChR
Pilocarpine nitrate
Cat.No: T1231
Synonym: 匹鲁卡品硝酸盐,Pilagan,硝酸毛果芸香碱,Pilofrin
Target: AChR
TargetMol Loading
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