Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T63115 |
Perphenazine dihydrochloride
|
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Perphenazine dihydrochloride 是一种口服具有活力的多巴胺受体 (dopamine receptor) 和组胺-1 受体 (histamine-1 receptor) 拮抗剂,作用于 D2 (Ki: 0.56 nM)、D3 (Ki: 0.43 nM)、5-HT2A (Ki: 0.6 nM)。Perphenazine dihydrochloride 也能够结合 Alpha-1A 肾上腺素受体。Perphenazine dihydrochloride 能够诱导细胞凋亡,并抑制癌细胞增殖。Perphenazine dihydrochloride 能够用于研究精神疾病、癌症、炎症。 | |||
T12411 |
Perphenazine D8 Dihydrochloride
|
Others | Others |
Perphenazine D8 Dihydrochloride is the deuterium labeled Perphenazine, which is an antipsychotic drug. |