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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22393 Palonosetron

RS25259,帕洛诺司琼,RS 25259 197

5-HT Receptor GPCR/G Protein; Neuroscience
Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).
T37246 Palonosetron N-oxide

Palonosetron N-oxide is a metabolite of the serotonin (5-HT) receptor subtype 5-HT3antagonist palonosetron .1It is also a potential impurity in palonosetron preparations.2Palonosetron N-oxide is a degradation product formed by exposure to oxidative stress. 1.Stoltz, R.A., Cyong, J.-C., Shah, A., et al.Pharmacokinetic and safety evaluation of palonosetron, a 5-hydroxytryptamine-3 receptor antagonist, in U.S. and Japanese healthy subjectsJ. Clin. Pharmacol.44(5)520-531(2004) 2.Vishnu Murthy, M., S...
T13437 (R,R)-Palonosetron Hydrochloride

Others Others
(R,R)-Palonosetron Hydrochloride is the active enantiomer of Palonosetron

化合物

Palonosetron
Cat.No: T22393
Synonym: RS25259,帕洛诺司琼,RS 25259 197
Target: 5-HT Receptor
Palonosetron N-oxide
Cat.No: T37246
Synonym:
Target:
(R,R)-Palonosetron Hydrochloride
Cat.No: T13437
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1156 Palonosetron hydrochloride

盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259

5-HT Receptor GPCR/G Protein; Neuroscience
Palonosetron hydrochloride (RS 25259) 是一种 5-HT3 拮抗剂,用于预防和治疗化疗引起的恶心和呕吐。

天然产物

Palonosetron hydrochloride
Cat.No: T1156
Synonym: 盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259
Target: 5-HT Receptor
TargetMol Loading
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