购物车

搜索结果

Search Results for " pwwp1 "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T8879 MR837

ZINC30303842,NSD2-PWWP1 antagonist 3f

Others; Histone Methyltransferase Chromatin/Epigenetic; Others
MR837 (NSD2-PWWP1 antagonist 3f) 是可与人核受体结合 SET 结构域蛋白(PWWP 结构域) 结合的NSD2-PWWP1抑制剂。
T9584 UNC6934

Others; Histone Methyltransferase Chromatin/Epigenetic; Others
UNC6934 是一种针对 NSD2 的 N 端 PWWP (PWWP1) 结构域的化学探针,可定位核仁。
T10538 BI-9321

Others Others
BI-9321 is a selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist (Kd: 166 nM). BI-9321 is inactive against NSD2-PWWP1 and NSD3-PWWP2.
T10538L BI-9321 trihydrochloride

Others Others
BI-9321 trihydrochloride is a selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist (Kd: 166 nM). BI-9321 is inactive against NSD2-PWWP1 and NSD3-PWWP2.
T62705 NSD2-IN-1

NSD2-IN-1 (compound 38) 是一种有效的、高选择性的 NSD2-PWWP1(核受体结合 SET 结构域 2-PWWP1) 抑制剂,IC50为 0.11 μM。NSD2-IN-1 可以与 NSD2-PWWP1 结合,进而影响受 NSD2 调控的基因表达。NSD2-IN-1 可以诱导细胞凋亡 (apoptosis) 和细胞周期阻滞。
T79616 UNC7096

Histone Methyltransferase Chromatin/Epigenetic
UNC7096为一种选择性NSD2-PWWP1抑制剂,其Kd为46 nM,拥有潜在治疗NSD2相关疾病的能力。
T79615 MS9715

Histone Methyltransferase Chromatin/Epigenetic
MS9715是一高效的选择性NSD3PROTAC,通过E3连结酶VHL配体与NSD3的PWWP1结构域相结合而由BI-9321设计。该化合物对于NSD3依赖性癌症治疗的研究具有潜在应用价值。

化合物

MR837
Cat.No: T8879
Synonym: ZINC30303842,NSD2-PWWP1 antagonist 3f
Target: Others, Histone Methyltransferase
UNC6934
Cat.No: T9584
Synonym:
Target: Others, Histone Methyltransferase
BI-9321
Cat.No: T10538
Synonym:
Target: Others
BI-9321 trihydrochloride
Cat.No: T10538L
Synonym:
Target: Others
NSD2-IN-1
Cat.No: T62705
Synonym:
Target:
UNC7096
Cat.No: T79616
Synonym:
Target: Histone Methyltransferase
MS9715
Cat.No: T79615
Synonym:
Target: Histone Methyltransferase
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼