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6

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8552 PSEM 89S TFA

AChR Neuroscience
PSEM 89S TFA 是一种脑渗透性和选择性离子通道激动剂,分别对 Q79G 和 L141F 具有正交选择性。
T28460 Psammaplysene B

Psammaplysene B is a FOXO1a nuclear export inhibitor.
T28459 Psammaplysene A

Psammaplysene A is a FOXO1a nuclear export inhibitor.
T124402 7-O-Acetyllycopsamine N-oxide

7-O-Acetyllycopsamine N-oxide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124402。
T123864 Lycopsamine N-oxide

Lycopsamine N-oxide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T123864。
T37391 PSEM 308 hydrochloride

PSAM (pharmacologically selective actuator module) agonist. Activates PSAML141F-GlyR chimeric ion channels. Inhibits activity of neurons expressing PSAML141F-GlyR in vivo and activates locus coeruleus noradrenergic neurons expressing PSAML141F,Y115F-5-HT3 ion channels. Recommended concentration for use in mice is 5 mg/kg or lower. Plasmid vectors for the transfection of cells with PSAML141F-GlyR and PSAML141F,Y115F-5-HT3 are available from Addgene. Lovett-Barron et al (2012) Regulation of neu...

化合物

PSEM 89S TFA
Cat.No: T8552
Synonym:
Target: AChR
Psammaplysene B
Cat.No: T28460
Synonym:
Target:
Psammaplysene A
Cat.No: T28459
Synonym:
Target:
7-O-Acetyllycopsamine N-oxide
Cat.No: T124402
Synonym:
Target:
Lycopsamine N-oxide
Cat.No: T123864
Synonym:
Target:
PSEM 308 hydrochloride
Cat.No: T37391
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T33029 7-Acetyllycopsamine

Lycopsamine `1-acetate,7-乙酰基环磷酰胺

Lycopsamine `1-acetate is a bioactive chemical.
T36303 Psammaplin A

Psammaplin A, a marine metabolite, functions as a robust inhibitor of HDAC and DNA methyltransferases, displaying notable potency and selectivity as a DAC1 inhibitor, with an IC50 value of 0.9 nM. It exhibits antimicrobial effects against Gram-positive bacteria and inhibits both DNA synthesis and DNA gyrase activity, also demonstrating antitumor activity[1][2].
T33028 Lycopsamine

Lycopsamine is a bioactive chemical.

天然产物

7-Acetyllycopsamine
Cat.No: T33029
Synonym: Lycopsamine `1-acetate,7-乙酰基环磷酰胺
Target:
Psammaplin A
Cat.No: T36303
Synonym:
Target:
Lycopsamine
Cat.No: T33028
Synonym:
Target:
TargetMol Loading
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