Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79144 |
PROTAC MEK1 Degrader-1
|
PROTACs | PROTAC |
PROTACMEK1Degrader-1是一种针对MEK1的PROTAC,显示出pIC50值为7.0。该化合物由MEK1抑制剂与von Hippel-Lindau配体构成,能够抑制ERK1/2的磷酸化,并对A375细胞展现出抗增殖活性。 |