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Cat. No. Product Name Target Signaling Pathways
T16667 PROTAC Sirt2 Degrader-1

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
PROTAC Sirt2 Degrader-1 is a SirReal-based PROTAC, acts as a Sirt2 degrader, composed of a highly potent and isotype-selective Sirt2 inhibitor, a linker, and a bona fide cereblon ligand for E3 ubiquitin ligase. PROTAC Sirt2 Degrader-1 shows an IC50 of 0.25 μM for Sirt2, with no effect on Sirt1/Sirt3 (IC50s > 100 μM)[1].

化合物

PROTAC Sirt2 Degrader-1
Cat.No: T16667
Synonym:
Target: Sirtuin
TargetMol Loading
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