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Cat. No. Product Name Target Signaling Pathways
T17728 PROTAC CDK9 degrader-2

Others Others
PROTAC CDK9 degrader-2 (compounds 11c) is a potent and selective CDK9 degrader based on PROTAC, with an IC50 of 17 μM in MCF-7 cell lines. Natural product Wogonin binds ubiquitin E3 ligase cereblon (CRBN) via a linker to form PROTAC[1].
T79904 PROTAC CDK9/CycT1 Degrader-2

CDK Cell Cycle/Checkpoint
PROTACCDK9/CycT1 Degrader-2CDK9表现出较高的抑制效能,具有一个IC50值为45 nM。
T10742 CDK9-IN-10

CDK Cell Cycle/Checkpoint
CDK9-IN-10 是一种有效的 CDK9 抑制剂。CDK9-IN-10 是 PROTAC CDK9 degrader-2 的配体。

化合物

PROTAC CDK9 degrader-2
Cat.No: T17728
Synonym:
Target: Others
PROTAC CDK9/CycT1 Degrader-2
Cat.No: T79904
Synonym:
Target: CDK
CDK9-IN-10
Cat.No: T10742
Synonym:
Target: CDK
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