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Cat. No. Product Name Target Signaling Pathways
T12552 PROTAC CDK2/9 Degrader-1

CDK Cell Cycle/Checkpoint
PROTAC CDK2/9 Degrader-1 is a potent CDK2 and CDK9 dual degrader(DC50 of 62 nM and 33 nM).
T17728 PROTAC CDK9 degrader-2

Others Others
PROTAC CDK9 degrader-2 (compounds 11c) is a potent and selective CDK9 degrader based on PROTAC, with an IC50 of 17 μM in MCF-7 cell lines. Natural product Wogonin binds ubiquitin E3 ligase cereblon (CRBN) via a linker to form PROTAC[1].

化合物

PROTAC CDK2/9 Degrader-1
Cat.No: T12552
Synonym:
Target: CDK
PROTAC CDK9 degrader-2
Cat.No: T17728
Synonym:
Target: Others
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