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Cat. No. Product Name Target Signaling Pathways
T74138 PROTAC Bcl-xL degrader-2

PROTACs PROTAC
PROTACBcl-xLdegrader-2 是一种基于von Hippel-Lindau 配体的Bcl-xL(Bcl-2家族成员) 降解剂,IC50为 0.6 nM。
T39910 Desmorpholinyl Navitoclax-NH-Me

Desmorpholinyl ABT-263-NH-Me,Desmorpholinyl Navitoclax-NH-Me

BCL Apoptosis
Desmorpholinyl Navitoclax-NH-Me (Desmorpholinyl ABT-263-NH-Me) is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739, a PROTAC BCL-XL degrader [1] [2].
T40135 PZ703b

PROTACs PROTAC
PZ703b is a novel BCL-XL PROTAC degrader with enhanced BCL-2 inhibition.
T73957 PROTAC Bcl-xL degrader-1

PROTACBcl-xL degrader-1是一种针对Bcl-xLBcl-2家族成员)的PROTAC,具备配体结合基团、linker以及IAPE3连接酶结合基团。这种化合物是一个有效的Bcl-xL降解剂,对人血小板和MyLa 1929细胞显示出明显的毒性,其IC50值分别为62 nM和8.5 μM。
T39909 XZ739

XZ739

PROTACs PROTAC
XZ739 is a Cereblon-dependent PROTAC BCL-XL degrader, targeting a member of the Bcl-2 family, with a DC50 value of 2.5 nM in MOLT-4 cells after 16 hours of treatment. Additionally, XZ739 elicits cell death via caspase-mediated apoptosis.
T73826 PZ703b hydrochloride

PROTACs PROTAC
PZ703b hydrochloride 是一种Bcl-xlPROTAC 降解剂,可以诱导细胞凋亡 (apoptosis),抑制癌细胞增殖。PZ703b hydrochloride 可用于膀胱癌的研究。

化合物

PROTAC Bcl-xL degrader-2
Cat.No: T74138
Synonym:
Target: PROTACs
Desmorpholinyl Navitoclax-NH-Me
Cat.No: T39910
Synonym: Desmorpholinyl ABT-263-NH-Me,Desmorpholinyl Navitoclax-NH-Me
Target: BCL
PZ703b
Cat.No: T40135
Synonym:
Target: PROTACs
PROTAC Bcl-xL degrader-1
Cat.No: T73957
Synonym:
Target:
XZ739
Cat.No: T39909
Synonym: XZ739
Target: PROTACs
PZ703b hydrochloride
Cat.No: T73826
Synonym:
Target: PROTACs
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