Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12560 |
PROTAC BRD9 Degrader-1
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
PROTAC BRD9 Degrader-1 is a lead PROTAC BRD9 chemical degrader with IC50 of 13.5 nM. | |||
T77975 |
PROTAC BRD9 Degrader-6
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
PROTACBRD9Degrader-6,作为BRD9降解剂,表现出高效率(IC50=0.13 nM),主要应用于BAF复合物相关疾病的研究领域。 | |||
T81382 | PROTAC BRD9 Degrader-7 | PROTACs | PROTAC |
PROTACBRD9Degrader-7 是具有口服活性的BRD9选择性降解剂,DC50 值为 1.02 nM,表现出较好的口服生物利用度,其Cmax 达到 3436.95 ng/mL。 |