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Cat. No.	Product Name	Target	Signaling Pathways
T62581	PPARγ agonist 6
	PPARγ agonist 6 (Compound 12) 是一种选择性 PPARγ 的有效激动剂。PPARγ agonist 6 具有潜力进行癌症疾病的研究。
T15453	GW7647 2-[[4-[2-[[环己基氨基)羰基](4-环己基丁基)氨基]乙基]苯基]硫基]-2-甲基丙酸	PPAR	DNA Damage/DNA Repair; Metabolism
	GW7647 是一种PPARα有效激动剂，对人 PPARα、PPARγ 和 PPARδ 的EC50值分别为 6、1.1 和 6.2 μM。
T7159	L-165041	PPAR	DNA Damage/DNA Repair; Metabolism
	L-165041 是一种细胞渗透性 PPARδ激动剂，可在 NIH-PPARδ 细胞中诱导脂肪细胞分化，对 PPARδ 和 PPARγ 的 Ki 值分别为 6 nM 和约 730 nM。
T35638	SR 1903
	SR 1903 is a modulator of retinoic acid receptor-related orphan receptor γ (RORγ) and liver X receptor (LXR).1 It is an inverse agonist of RORγ (IC50 = ~100 nM in a cell-based reporter assay) and an agonist of LXR. It also binds to peroxisome proliferator-activated receptor γ (PPARγ; IC50 = 209 nM) but does not activate it. SR 1903 (10 μM) inhibits LPS-induced expression of triggering receptor expressed on myeloid cells 1 (TREM-1) in RAW 264.7 cells. It also inhibits LPS-induced expression of th...
T35468	(±)19(20)-EDP Ethanolamide
	(±)19(20)-EDP ethanolamide is an ω-3 endocannabinoid epoxide and cannabinoid (CB) receptor agonist (EC50s = 108 and 280 nM for CB1 and CB2, respectively). It is produced through direct epoxygenation of docosahexaenoyl ethanolamide by cytochrome P450 (CYP) epoxygenases. (±)19(20)-EDP ethanolamide (25 μM) reduces the viability of 143B metastatic osteosarcoma cells. It decreases the production of IL-6 and increases the production of IL-10 when used at concentrations ranging from 2.5 to 10 μM in BV-...